COMT
Entacapone CAS No. 130929-57-6
Entacapone is definitely a critical, reversible catechol-O-methyl transferase (COMT) inhibitor with IC50 of 151 nM.
GABAAR
Dihydromyricetin CAS No. 27200-12-0
Dihydromyricetin (Ampelopsin, Ampeloptin) is surely a all-all-natural antioxidant flavonoid from Ampelopsis grossedentata.
5-HT1D
LY310762 CAS No. 192927-92-7
LY310762 is really a 5-HT1D receptor antagonist with Ki of 249 nM, simply by using a vulnerable affinity for five-HT1B receptor.
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